H. Elokdah : rechercher sur Z-Library

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1

ChemInform Abstract: Effects of 2-(Substituted-sulfanyl)-3,5-dihydro-imidazole-4-one (V) and 2-(Substituted-sulfanyl)-1H-imidazole-4,5-dione Derivatives (VIII) on Serum HDL-Cholesterol.

Hassan Elokdah, Theodore Sulkowski, David Cochran, Mar-Lee McKean, Elaine Quinet

Journal:

Année:

2000

Fichier:

PDF, 31 KB

2000

2

ChemInform Abstract: Design and Synthesis of Tricyclic Derivatives as High Density Lipoprotein Cholesterol Enhancers.

Hassan Elokdah, Sie-Yearl Chai, Douglas Ho, Theodore Sulkowski

Journal:

Année:

2001

Fichier:

PDF, 29 KB

2001

3

Novel Human Metabolites of the Angiotensin-II Antagonist Tasosartan and Their Pharmacological Effects.

Hassan M. Elokdah, Gregory S. Friedrichs, Sie-Yearl Chai, Boyd L. Harrison, John Primeau, Michael Chlenov, David L. Crandall

Journal:

Année:

2002

Fichier:

PDF, 29 KB

2002

4

Tiplaxtinin, a Novel, Orally Efficacious Inhibitor of Plasminogen Activator Inhibitor-1: Design, Synthesis, and Preclinical Characterization.

Hassan Elokdah, Magid Abou-Gharbia, James K. Hennan, Geraldine McFarlane, Cheryl P. Mugford, Girija Krishnamurthy, David L. Crandall

Journal:

Année:

2004

Fichier:

PDF, 11 KB

2004

5

Novel 1-(azacyclyl)-3-arylsulfonyl-1H-pyrrolo[2,3-b]pyridines as 5-HT6 agonists and antagonists

Hassan Elokdah, David Li, Geraldine McFarlane, Ronald C. Bernotas, Albert J. Robichaud, Ronald L. Magolda, Guo Ming Zhang, Deborah Smith, Lee E. Schechter

Journal:

Bioorganic & Medicinal Chemistry

Année:

2007

Langue:

english

Fichier:

PDF, 327 KB

english, 2007

6

Regioselective Suzuki coupling of benzofuran or benzothiophene boronic acids and dibromo substituted naphthalenes: synthesis of a potent inhibitor of plasminogen activator inhibitor-1

Zheng Wang, Hassan Elokdah, Geraldine McFarlane, Sherry Pan, Madelene Antane

Journal:

Tetrahedron Letters

Année:

2006

Langue:

english

Fichier:

PDF, 127 KB

english, 2006

7

Efficient one-pot synthesis of substituted 2-amino-1,3,4-oxadiazoles

Eugene L. Piatnitski Chekler, Hassan M. Elokdah, John Butera

Journal:

Tetrahedron Letters

Année:

2008

Langue:

english

Fichier:

PDF, 144 KB

english, 2008

8

Effects of 2-(substituted-sulfanyl)-3,5-dihydro-imidazole-4-one and 2-(substituted-sulfanyl)-1H-imidazole-4,5-dione derivatives on serum HDL-cholesterol

Hassan Elokdah, Theodore Sulkowski, David Cochran, Mar-Lee McKean, Elaine Quinet

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2000

Langue:

english

Fichier:

PDF, 181 KB

english, 2000

9

Design and synthesis of tricyclic derivatives as high density lipoprotein cholesterol enhancers

Hassan Elokdah, Sie-Yearl Chai, Douglas Ho, Theodore Sulkowski

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2001

Langue:

english

Fichier:

PDF, 230 KB

english, 2001

10

Novel human metabolites of the angiotensin-II antagonist tasosartan and their pharmacological effects

Hassan M Elokdah, Gregory S Friedrichs, Sie-Yearl Chai, Boyd L Harrison, John Primeau, Michael Chlenov, David L Crandall

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2002

Langue:

english

Fichier:

PDF, 194 KB

english, 2002

11

Characterization and comparative evaluation of a structurally unique PAI-1 inhibitor exhibiting oral in-vivo efficacy

D. L. Crandall, H. Elokdah, L. Di, J. K. Hennan, N. V. Gorlatova, D. A. Lawrence

Journal:

Journal of Thrombosis and Haemostasis

Année:

2004

Langue:

english

Fichier:

PDF, 195 KB

english, 2004

12

WAY-140312 reduces plasma PAI-1 while maintaining normal platelet aggregation

David L Crandall, James K Hennan, Hassan Elokdah, Girija Krishnamurthy, Thomas M Antrilli, Jean S Bauer, Gwen A Morgan, Robert E Swillo

Journal:

Biochemical and Biophysical Research Communications

Année:

2003

Langue:

english

Fichier:

PDF, 222 KB

english, 2003

13

Design, Synthesis, and Biological Evaluation of Thio-Containing Compounds with Serum HDL-Cholesterol-Elevating Properties

Elokdah, Hassan, Sulkowski, Theodore S., Abou-Gharbia, Magid, Butera, John A., Chai, Sie-Yearl, McFarlane, Geraldine R., McKean, Mar-Lee, Babiak, John L., Adelman, Steven J., Quinet, Elaine M.

Journal:

Journal of Medicinal Chemistry

Année:

2004

Langue:

english

Fichier:

PDF, 183 KB

english, 2004

14

Tiplaxtinin, a Novel, Orally Efficacious Inhibitor of Plasminogen Activator Inhibitor-1: Design, Synthesis, and Preclinical Characterization

Elokdah, Hassan, Abou-Gharbia, Magid, Hennan, James K., McFarlane, Geraldine, Mugford, Cheryl P., Krishnamurthy, Girija, Crandall, David L.

Journal:

Journal of Medicinal Chemistry

Année:

2004

Langue:

english

Fichier:

PDF, 66 KB

english, 2004

15

Mechanism of Inactivation of Plasminogen Activator Inhibitor-1 by a Small Molecule Inhibitor

Gorlatova, N. V., Cale, J. M., Elokdah, H., Li, D., Fan, K., Warnock, M., Crandall, D. L., Lawrence, D. A.

Journal:

Journal of Biological Chemistry

Année:

2007

Langue:

english

Fichier:

PDF, 940 KB

english, 2007

16

Enhanced clearance of A in brain by sustaining the plasmin proteolysis cascade

Jacobsen, J. S., Comery, T. A., Martone, R. L., Elokdah, H., Crandall, D. L., Oganesian, A., Aschmies, S., Kirksey, Y., Gonzales, C., Xu, J., Zhou, H., Atchison, K., Wagner, E., Zaleska, M. M., Das, I

Journal:

Proceedings of the National Academy of Sciences

Année:

2008

Langue:

english

Fichier:

PDF, 866 KB

english, 2008

17

Neutralization of Plasminogen Activator Inhibitor I (PAI-1) by the Synthetic Antagonist PAI-749 via a Dual Mechanism of Action

Gardell, S. J., Krueger, J. A., Antrilli, T. A., Elokdah, H., Mayer, S., Orcutt, S. J., Crandall, D. L., Vlasuk, G. P.

Journal:

Molecular Pharmacology

Année:

2007

Langue:

english

Fichier:

PDF, 368 KB

english, 2007

18

ID: 225 Mechanistic Studies on the Inactivation of Plasminogen Activator Inhibitor (PAI-1) by PAI-749, a Small Molecule PAI-1 Antagonist

Gardell, S., Antrilli, T., Elokdah, H., Krueger, J., Mayer, S., Orcutt, S., Vlasuk, G., Crandall, D.

Journal:

Journal of Thrombosis and Haemostasis

Année:

2006

Langue:

english

Fichier:

PDF, 220 KB

english, 2006

19

Mapping of a Conformational Epitope on Plasminogen Activator Inhibitor-1 by Random Mutagenesis: IMPLICATIONS FOR SERPIN FUNCTION

Gorlatova, N. V., Elokdah, H., Fan, K., Crandall, D. L., Lawrence, D. A.

Journal:

Journal of Biological Chemistry

Année:

2003

Langue:

english

Fichier:

PDF, 994 KB

english, 2003

20

Dose-dependent thrombus resolution due to oral plasminogen activator inhibitor (PAI)-1 inhibition with tiplaxtinin in a rat stenosis model of venous thrombosis

Baxi, Sanjiv, Crandall, David, Meier, Thomas, Wrobleski, Shirley, Hawley, Angela, Farris, Diana, Elokdah, Hassan, Sigler, Robert, Schaub, Robert, Wakefield, Thomas, Myers, Daniel

Journal:

Thrombosis and Haemostasis

Année:

2008

Fichier:

PDF, 298 KB

2008